您的位置: 首页 > 农业专利 > 详情页

PRODRUG OF FLUORINE-CONTAINING AMINO ACID
专利权人:
TAISHO PHARMACEUTICAL CO.; LTD.
发明人:
HASHIHAYATA, TAKASHI,OTAKE, NORIKAZU,MIYAKOSHI, NAOKI,SAKAGAMI, KAZUNARI
申请号:
RSP20170883
公开号:
RS56328B1
申请日:
2013.05.31
申请国别(地区):
RS
年份:
2017
代理人:
摘要:
Provided are a fluorine-containing amino acid prodrug represented by general formula (I) that makes a fluorine-containing amino acid which is a group 2 metabotropic glutamate receptor agonist into a prodrug, or a pharmaceutically acceptable salt thereof. More specifically, provided is a prodrug that increases the in vivo exposure and enhances the oral absorbability and other mucosal absorbability of a parent compound that acts on group 2 metabotropic glutamate receptors as an agent for the treatment or prevention of diseases in which group 2 metabotropic glutamate receptors are said to be involved, such as: schizophrenia, anxiety disorder and its related diseases, depression, bipolar disorder, epilepsy, developmental disorders, sleep disorders, and other neuropsychiatric diseases and drug dependence, cognitive disorders, Alzheimers disease, Huntingtons chorea, Parkinsons disease, movement disorders associated with muscular rigidity, cerebral ischemia, cerebral insufficiency, spinal cord disorders, cephalopathy, and other neurological diseases.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充