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GPR119 receptor modulators and the treatment of disorders related to this
- 专利权人:
- ARENA PHARMACEUTICALS; INC.
- 发明人:
- JONES, ROBERT M.,LEHMANN, JUERG,CHEN, WEICHAO,EDWARDS, JEFFREY,MARQUEZ, GLEN,MORGAN, MICHAEL E.,SADEQUE, ABU J.M.,KIM, SUN HEE
- 申请号:
- CR20130145
- 公开号:
- CR20130145A
- 申请日:
- 2013.03.22
- 申请国别(地区):
- CR
- 年份:
- 2013
- 代理人:
- 摘要:
- The present Invention relates to 5 GPR119 receptor agonists: 3-fluoro-4 - (4-fluoro-6 - 5 - (4 - (3 - (2 - fluoropropan - 2 - il) - 1,2,4 - Oxadiazoles - 5 - il) piperidin-1-yl) - 4 - ilamino pyrimidin-2-yl) - n, n-dimethylbenzamide; 3 - 4 - 5 - fluoro - (4-fluoro-6 - (4 - (3 - (2 - fluoropropan - 2 - il) - 1,2,4 - Oxadiazoles - 5 - il) piperidin-1-yl) pirimidi 4 -) - N - ilamino n-methylbenzamide; y10 3-fluoro-4 - (4-fluoro-6 - 5 - (4 - (3 - (2 - fluoropropan - 2 - 1.2, - il)Oxadiazoles - 4 - 5 - il) piperidin-1-yl) pyrimidin-2-yl) - 4 - ilamino benzamide, and pharmaceutically acceptable salts, solvates and hydrates of theseLa presente invención se refiere a los agonistas del receptor 5 GPR119:3-fluoro-4-(5-fluoro-6-(4-(3-(2-fluoropropan-2-il)-1,2,4-oxadiazol-5-il)piperidin-1- il)pirimidin-4-ilamino)-N,N-dimetilbenzamida; 3-fluoro-4-(5-fluoro-6-(4-(3-(2-fluoropropan-2-il)-1,2,4-oxadiazol-5- il)piperidin-1-il)pirimidin-4-ilamino)-N-metilbenzamida; y10 3-fluoro-4-(5-fluoro-6-(4-(3-(2-fluoropropan-2-il)-1,2,4-oxadiazol-5-il)piperidin-1-il)pirimidin-4- ilamino)benzamida, y a sales, solvatos e hidratos farmacéuticamente aceptables de estos
- 来源网站:
- 中国工程科技知识中心
- 来源网址:
- http://www.ckcest.cn/home/