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GPR119 receptor modulators and the treatment of disorders related to this
专利权人:
ARENA PHARMACEUTICALS; INC.
发明人:
JONES, ROBERT M.,LEHMANN, JUERG,CHEN, WEICHAO,EDWARDS, JEFFREY,MARQUEZ, GLEN,MORGAN, MICHAEL E.,SADEQUE, ABU J.M.,KIM, SUN HEE
申请号:
CR20130145
公开号:
CR20130145A
申请日:
2013.03.22
申请国别(地区):
CR
年份:
2013
代理人:
摘要:
The present Invention relates to 5 GPR119 receptor agonists: 3-fluoro-4 - (4-fluoro-6 - 5 - (4 - (3 - (2 - fluoropropan - 2 - il) - 1,2,4 - Oxadiazoles - 5 - il) piperidin-1-yl) - 4 - ilamino pyrimidin-2-yl) - n, n-dimethylbenzamide; 3 - 4 - 5 - fluoro - (4-fluoro-6 - (4 - (3 - (2 - fluoropropan - 2 - il) - 1,2,4 - Oxadiazoles - 5 - il) piperidin-1-yl) pirimidi 4 -) - N - ilamino n-methylbenzamide; y10 3-fluoro-4 - (4-fluoro-6 - 5 - (4 - (3 - (2 - fluoropropan - 2 - 1.2, - il)Oxadiazoles - 4 - 5 - il) piperidin-1-yl) pyrimidin-2-yl) - 4 - ilamino benzamide, and pharmaceutically acceptable salts, solvates and hydrates of theseLa presente invención se refiere a los agonistas del receptor 5 GPR119:3-fluoro-4-(5-fluoro-6-(4-(3-(2-fluoropropan-2-il)-1,2,4-oxadiazol-5-il)piperidin-1- il)pirimidin-4-ilamino)-N,N-dimetilbenzamida; 3-fluoro-4-(5-fluoro-6-(4-(3-(2-fluoropropan-2-il)-1,2,4-oxadiazol-5- il)piperidin-1-il)pirimidin-4-ilamino)-N-metilbenzamida; y10 3-fluoro-4-(5-fluoro-6-(4-(3-(2-fluoropropan-2-il)-1,2,4-oxadiazol-5-il)piperidin-1-il)pirimidin-4- ilamino)benzamida, y a sales, solvatos e hidratos farmacéuticamente aceptables de estos
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