Lysine-based prodrugs of aspartyl protease inhibitors and processes for their preparation

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专利权人:

Guy Milot

发明人:

Guy Milot,Stephane Branchaud,Brent R. Stranix

申请号：

US12086184

公开号：

US08227450B2

申请日:

2006.11.30

申请国别(地区):

US

年份:

2012

代理人:

摘要：

The present invention provides processes for synthesizing lysine based compounds of the formulawherein R1 may be, for example, (HO)2P(O)—, (NaO)2P(O)—, wherein X may be, for example, NH2, Y may be H, F, Cl, or Br, and wherein n, X′, Y′, R2, R3, R4, R5 and R6 are as defined herein.

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