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1H-indazol-3-karboksamidne spojine kot inhibitorji glikogen sintaza-kinaze-3beta
专利权人:
AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO - A.C.R.A.F. - S.P.A
发明人:
ALISI MARIA ALESSANDRA,CAZZOLLA NICOLA,DRAGONE PATRIZIA,FURLOTTI GUIDO,MAUGERI CATERINA,OMBRATO ROSELLA,MANCINI FRANCESCA,ALISI Maria Alessandra,CAZZOLLA Nicola,DRAGONE Patrizia,FURLOTTI Guido,MAUGERI Caterina,OMBRATO
申请号:
SI201330134
公开号:
SI2817302T1
申请日:
2013.02.07
申请国别(地区):
SI
年份:
2016
代理人:
摘要:
The present invention relates to the 1H-indazole-3-carboxamide compounds having the following general formula (I) as glycogen synthase kinase 3 beta (GSK-3&bgr;) inhibitors and to their use in the treatment of GSK-3p-related disorders such as, for example, (i) insulin-resistance disorders; (ii) neurodegenerative diseases; (iii) mood disorders; (iv) schizophrenic disorders; (v) cancerous disorders; (vi) inflammation, (vii) substance abuse disorders; (viii) epilepsies; and (ix) neuropathic pain.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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