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3,5,5-trimethyl-2 - [5 - (2-phenyl-phenyl) - 2-pyridyl / pyridinediol] pyridan-4-one, glutamate metabolizing receptor antagonist; preparation procedure; drug synthesis containing these substances; used in the treatment of anxiety, pain, depression, Parkinson's disease, etc
专利权人:
F. HOFFMANN-LA ROCHE AG.
发明人:
JAESCHKE, GEORG,LINDEMANN, LOTHAR,RICCI, ANTONIO,STADLER, HEINZ,VIERA, ERIC,MARTIN, RAINER E.,RUENER, DANIEL
申请号:
CL2015003761
公开号:
CL2015003761A1
申请日:
2015.12.30
申请国别(地区):
CL
年份:
2016
代理人:
摘要:
<;p>; THE PRESENT INVENTION IS RELATED TO ETHINYL DERIVATIVES FROM FOAcute; RMULA I: IN WHICH: Y IS NOT CH, R1 IS HYDROacute; GENE, FLUUTE OR CHLORINE, AND R2 IS HYDROacute; GENE OR METHYL, OR A PHARMACEUTICALLY ACCEPTABLE ADDITIONAL SALT OF PHARMACEUTICALLY ACCEPTABLE AS GLUTAMATE METABOTROPIC RECIPIENT ANTAGONISTS; PREPARATION PROCEDURE; PHARMACEUTICAL COMPOSITION THAT UNDERSTANDS THEM; AND ITS USE FOR THE TREATMENT OF ANXIETY, PAIN, DEPRESSION, PARKINSON'S DISEASE, AMONG OTHERS. <;/p>;<;p>;LA PRESENTE INVENCIÓ;N SE REFIERE A DERIVADOS DE ETINILO DE FÓ;RMULA I: EN LA QUE: Y ES N O CH, R1 ES HIDRÓ;GENO, FLÚ;OR O CLORO, Y R2 ES HIDRÓ;GENO O METILO, O UNA SAL DE ADICIÓ;N DE Á;CIDO FARMACÉ;UTICAMENTE ACEPTABLE DE LOS MISMOS, COMO ANTAGONISTAS DE RECEPTOR METABOTRÓ;PICO DE GLUTAMATO; PROCEDIMIENTO DE PREPARACIÓ;N; COMPOSICIÓ;N FARMACÉ;UTICA QUE LOS COMPRENDE; Y SU USO PARA EL TRATAMIENTO DE LA ANSIEDAD, DOLOR, DEPRESIÓ;N, ENFERMEDAD DE PARKINSON, ENTRE OTRAS.<;/p>;
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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