GENENTECH, INC.;Constellation Pharmaceuticals, Inc.
发明人:
申请号:
EP19191423.3
公开号:
EP3632915A1
申请日:
2015.11.25
申请国别(地区):
EP
年份:
2020
代理人:
摘要:
The present invention relates to compounds of formula (I) or formula (II):and to salts thereof, wherein R1-R4 of formula (I) and R1-R3 of formula (II) have any of the values defined herein, and compositions and uses thereof. The compounds are useful as inhibitors of CBP and/or EP300. Also included are pharmaceutical compositions comprising a compound of formula (I) of formula (II) or a pharmaceutically acceptable salt thereof, and methods of using such compounds and salts in the treatment of various CBP and/or EP300-mediated disorders.