The present invention relates to a novel method for preparing a 1 oxacephalosporin derivative which is an intermediate for the synthesis of 1 oxacephalosporin which is useful as an antibacterial agent. The preparation method of the present invention uses a simple halogenating agent to show remarkable stability have a simple reaction process allow a reaction to be readily controlled and reduce reaction time and thus is very efficient and improves the production yield of 1 oxacephalosporin which is useful as an antibacterial agent.