CHRISTIAN HUBSCHWERLEN,PHILIPPE PANCHAUD,JEAN-LUC SPECKLIN
申请号:
MYPI 20091893
公开号:
MY148847A
申请日:
2007.11.09
申请国别(地区):
MY
年份:
2013
代理人:
摘要:
THE INVENTION RELATES TO NOVEL CHIMERIC ANTIBIOTICS OF FORMULA I WHEREIN R¹ REPRESENTS OH, OPO₃H₂ OR OCOR⁵; R² REPRESENTS H, OH OR OPO₃H₂; A REPRESENTS N OR CR⁶; R³ REPRESENTS H OR FLUORINE; R⁴IS H, (C₁-C₃) ALKYL, OR CYCLOALKYL; R⁵ IS THE RESIDUE OF A NATURALLY OCCURRING AMINO ACID, OF THE ENANTIOMER OF A NATURALLY OCCURRING AMINO ACID OR OF DIMETHYLAMINOGLYCINE; R⁶ REPRESENTS H, ALKOXY OR HALOGEN; AND N IS 0 OR 1; AND TO SALTS (IN PARTICULAR PHARMACEUTICALLY ACCEPTABLE SALTS) OF COMPOUNDS OF FORMULA I. THESE CHIMERIC COMPOUNDS ARE USEFUL IN THE MANUFACTURE OF MEDICAMENTS FOR THE TREATMENT OF INFECTIONS (E.G. BACTERIAL INFECTIONS).