PEPTIDE EPOXYCETONES DESTINEES A L'INHIBITION DE PROTEASOME
- 专利权人:
- INC.;ONYX THERAPEUTICS
- 发明人:
- 申请号:
- EP07809745.8
- 公开号:
- EP2041158B1
- 申请日:
- 2007.06.19
- 申请国别(地区):
- EP
- 年份:
- 2013
- 代理人:
- 摘要:
- One aspect of the invention relates to inhibitors of formula (I) that preferentially inhibit immunoproteasome activity over constitutive proteasome activity. In certain embodiments, the invention relates to the treatment of immune related diseases, comprising administering a compound of the invention. In certain embodiments, the invention relates to the treatment of cancer, comprising administering a compound of the invention.
- 来源网站:
- 中国工程科技知识中心
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