您的位置: 首页 > 农业专利 > 详情页

Salts of pyrrolotriazine derivatives useful as TAM inhibitors
专利权人:
인사이트 코포레이션
发明人:
지아 중지앙,우 융중,판 융춘,저우 지아청,리 췬
申请号:
KR1020207012225
公开号:
KR1020200088308A
申请日:
2018.09.26
申请国别(地区):
KR
年份:
2020
代理人:
摘要:
N- (4-(4-amino-7-(1-isobutyrylpiperidin-4-yl)pyrrolo[1,2- f ][1,2,4]tri useful as an inhibitor of TAM kinase Azin-5-yl)phenyl)-1-isopropyl-2,4-dioxo-3-(pyridin-2-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide ( I) and N- (4-(4-amino-7-(1-isobutyrylpiperidin-4-yl)pyrrolo[1,2- f ][1,2,4]triazin-5-yl )Phenyl)-1-isopropyl-2,4-dioxo-3-phenyl-1,2,3,4-tetrahydropyrimidine-5-carboxamide (II) salt form, as well as related salt forms Methods and intermediates are provided. ,본원은 TAM 키나제의 억제제로서 유용한 N-(4-(4-아미노-7-(1-이소부티릴피페리딘-4-일)피롤로[1,2-f][1,2,4]트리아진-5-일)페닐)-1-이소프로필-2,4-디옥소-3-(피리딘-2-일)-1,2,3,4-테트라하이드로피리미딘-5-카복사미드 (I) 및 N-(4-(4-아미노-7-(1-이소부티릴피페리딘-4-일)피롤로[1,2-f][1,2,4]트리아진-5-일)페닐)-1-이소프로필-2,4-디옥소-3-페닐-1,2,3,4-테트라하이드로피리미딘-5-카복사미드(II)의 염 형태, 뿐만 아니라 그와 관련된 방법 및 중간체를 제공한다.,
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充