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dihydro-benzo oxazine and dihydro-pyrido oxazine derivatives
专利权人:
NOVARTIS AG
发明人:
ALEXANDER BAXTER SMITH,CHRISTOPH KALIS,FRÉDÉRIC ZECRI,GIORGIO CARAVATTI,HENRIK MOEBITZ,IAN LEWIS,KAREN KAMMERTOENS,KLEMENS HÖGENAUER,KONSTANZE HURTH,NICOLAS SOLDERMANN,PASCAL FURET,ROMAIN WOLF,SYLVIE
申请号:
BR112014015103
公开号:
BR112014015103A2
申请日:
2012.12.20
申请国别(地区):
BR
年份:
2017
代理人:
摘要:
patent summary: "dihydro-benzo-oxazine and dihydro-pyrido-oxazine derivatives". The invention relates to dihydro-benzo-oxazine and dihydro-pyrido-oxazine compounds of formula (I) and / or pharmaceutically acceptable salts and / or solvates thereof (i) wherein y, v, w , u, q, r1, r5, r7 and r30 are as defined in the description. Such compounds are suitable for treating a disease or disorder which is mediated by pi3k enzyme activity. 301resumo patente de invenção: "derivados de di-hidro-benzo-oxazina e di-hidro-pirido-oxazina". a invenção refere-se a compostos de di-hidro-benzo-oxazina e di-hidro-pirido-oxazina de fórmula (i) e/ou sais farmaceuticamente aceitáveis e/ou solvatos dos mesmos (i) em que y, v, w, u, q, r1, r5, r7 e r30 são conforme definidos na descrição. tais compostos são adequados para tratamento de uma doença ou distúrbio o qual é mediado por atividade de enzimas pi3k. 301
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