TRICYCLIC PYRAZOLOPYRIMIDINE DERIVATIVE

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专利权人:

发明人:

OHKI HITOSHI JAPAN,OKAYAMA TOORU JAPAN,IKEDA MASAHIRO JAPAN,OTA MASAHIRO JAPAN,SHIBATA YOSHIHIRO JAPAN,NAKANISHI TOSHIYUKI JAPAN,UEDA YASUSI JAPAN,SUZUKI NOBUYUKI JAPAN,MATUURA SHINJI JAPAN

申请号：

IN1696/MUMNP/2011

公开号：

IN2011MN01696A

申请日:

2011.08.16

申请国别(地区):

IN

年份:

2012

代理人:

摘要：

To provide a novel compound inhibiting the effect of HSP90, in particular a novel compound inhibiting the function of HSP90 as a chaperone protein and having antitumor activity. The present invention provides a pyrazolopyrimidine compound represented by formula (1) having various substituents which inhibits the ATPase activity of HSP90 and which has antitumor activity, an HSP90 inhibitor comprising a compound represented by formula (1), a medicament comprising a compound represented by formula (1), an anticancer agent comprising a compound represented by formula (1), a pharmaceutical composition comprising a compound represented by formula (1), and a method for treating cancer using a compound represented by formula (1).

来源网站：

中国工程科技知识中心

来源网址：

http://www.ckcest.cn/home/