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Highly water-soluble salts of a short acting phenylalkylamine calcium channel blocker and uses thereof
专利权人:
Milestone Pharmaceuticals Inc.
发明人:
MAGUIRE Martin P.
申请号:
MDE20180191
公开号:
MD3283067T2
申请日:
2016.04.13
申请国别(地区):
MD
年份:
2020
代理人:
摘要:
The invention refers to salts, which include a phenylalchilamine compound, which has a surprisingly high solubility in aqueous solution. The salts in this invention are recognised antagonists of L-type calcium channels and provide a new therapeutic platform for the treatment of cardiac arrhythmias such as paroxytic supraventricular tachycardia, stable angina and migraines.Invenţia se referă la săruri, care includ un compus fenilalchilamină, care prezintă o solubilitate surprinzător de mare în soluţie apoasă. Sărurile din prezenta invenţie sunt antagonişti recunoscuţi ai canalelor de calciu de tip L şi oferă o nouă platformă terapeutică pentru tratamentul aritmiilor cardiace, cum ar fi tahicardia supraventriculară paroxistică, angina stabilă şi migrenele.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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