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COMPOUND, DRUG, ANTIBACTERIAL AND THERAPEUTIC AGENTS FOR INFECTIONS, METHODS TO TREAT DISEASES AND INFECTIONS AND TO PRODUCE A DRUG, ANTIBACTERIAL AGENT AND THERAPEUTIC AGENT FOR INFECTIONS AND USE OF THE COMPOUND.
专利权人:
DAIICHI SANKYO COMPANY; LIMITED
发明人:
HISASHI TAKAHASHI,SATOSHI KOMORIYA,TAKAHIRO KITAMURA,TAKASHI ODAGIRI,HIROAKI INAGAKI,TOSHIFUMI TSUDA,KIYOSHI NAKAYAMA,MAKOTO TAKEMURA,KENICHI YOSHIDA,RIE MIYAUCHI,MASATOSHI NAGAMOCHI
申请号:
BRPI0720771
公开号:
BRPI0720771A2
申请日:
2007.12.28
申请国别(地区):
BR
年份:
2014
代理人:
摘要:
Intermediates of formula (Ia) or (Ib) are provided: wherein R 11 and R 21 represents a hydrogen atom or an amino-protecting group, and R 16 represents an amino-protecting group, useful for the production of quinolone synthetic antibacterial agent of formula (I) wherein substituents R 6 and R 7 taken together with the carbon atoms to which they are bonded form a cyclic structure which may contain an oxygen atom as a ring constituent atom, the cyclic structure forming a 5-4, 5-5, or 5-6 fused bicyclic pyrrolidinyl substituent, the substituent being bonded to a quinolone mother skeleton Q containing a pyridobenzoxazine structure:
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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