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PROCÉDÉ DEPRÉPARATION DE 4-AMINO-1- ((1S, 4R, 5S) -2-FLUORO-4,5-DIHYDROXY-3- HYDROXYMÉTHYL-CYCLOPENT-2-ENYL) -1H-PYRIMIDIN-2-ONE
专利权人:
Rexahn Pharmaceuticals; Inc.
发明人:
申请号:
EP16206409.1
公开号:
EP3246320A1
申请日:
2014.03.17
申请国别(地区):
EP
年份:
2017
代理人:
摘要:
Processes for the preparation of 4-amino-1-((1S,4R,5S)-2-fluoro-4,5-dihydroxy-3-hydroxymethyl-cyclopent-2-enyl)-1H-pyrimidin-2-one (13, RX-3117) and its intermediates are described.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/
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Process for the preparation of 4-amino-1 - ((1s, 4r, 5s) -2-fluoro-4,5-dihydroxy-3-hydroxymethyl-cyclopent-2-enii) -1h-pyrimidin-2-one
PROCEDE POUR LA PREPARATION DE 4-AMINO-1-((1S,4R,5S)-2-FLUORO-4,5-DIHYDROXY-3-HYDROXYMETHYL-CYCLOPENT-2-ENYL)-1H-PYRIMIDIN-2-ONE
Process for the preparation of 4-amino-1-((1S,4R,5S)-2-fluoro-4,5-dihydroxy-3-hydroxymethyl-cyclopent-2-enyl)-1H-pyrimidin-2-one
Process for the preparation of 4-amino-1-((1S,4R,5S)-2-fluoro-4,5-dihydroxy-3-hydroxymethyl-cyclopent-2-enyl)-1H-pyrimidin-2-one
Process for the preparation of 4-amino-1-((1S,4R, 5S)-2-fluoro-4,5-dihydroxy-3-hydroxymethyl-cyclopent-2-enyl)-1H-pyrimidin-2-one