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Synthetic rigidin analogues as anticancer agents, salts, solvates and prodrugs thereof, and method of producing same
专利权人:
发明人:
Igor V. Magedov,Snezna Rogelj,Liliya Vladlenovna Frolova,Alexander Vladimir Kornienko
申请号:
US13678987
公开号:
US08946246B2
申请日:
2012.11.16
申请国别(地区):
US
年份:
2015
代理人:
摘要:
A compound having the Formula I as follows:wherein R1 and R2 are selected from hydrogen, aryl, fused aryl, heteroaryl, saturated carbocylclic, partially saturated carbocyclic, saturated heterocyclic, partially saturated heterocyclic, C1-10 alkyl, haloalkyl, alkenyl, alkynyl, arylalkyl, arylalkenyl, arylalkynyl, heteroarylalkyl, heteroarylalkenyl, carbocycloalkyl, heterocycloalkyl, hydroxyalkyl, aminoalkyl, carboxyalkyl, nitroalkyl, cyanoalkyl, acetamidoalkyl, and acyloxyalkyl. A process for the preparation thereof is also provided.
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