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crystalline form 4 - ((r) -2 - {[6 - ((s) -3-methoxy-pyrrolidin-1-yl) -2-phenyl-pyrimidin-4-carbonyl] -amino} acid butyl ester hydrochloride -3-phosphono-propionyl) -piperazine-1-carboxylic acid process for preparing 4 - ((r) -2 - {[6 - ((s) -3-methoxy-pyrrolidin-1-butyl ester) hydrochloride yl) -2-phenyl-pyrimidine-4-carbonyl] -amino} -3-phosphono-propionyl) -piperazine-1-carboxylic acid pharmaceutical composition and 4 - ((r) -2 - {[6] butyl ester - ((s) -3-Methoxy-pyrrolidin-1-yl) -2-phenyl-pyrimidin-4-carbonyl] -amino} -3-phosphono-propionyl) -piperazine-1-carboxylic acid.
专利权人:
IDORSIA PHARMACEUTICALS LTD
发明人:
DANIEL LEUENBERGER,MARKUS VON RAUMER,STEFAN REBER
申请号:
BR112019004845
公开号:
BR112019004845A2
申请日:
2017.09.21
申请国别(地区):
BR
年份:
2019
代理人:
摘要:
The invention relates to crystalline forms of 4 - ((r) -2 - {[6 - ((s) -3-methoxy-pyrrolidin-1-yl) -2-phenyl-pyrimidine-2-butyl ester hydrochloride Carbonyl] amino} -3-phosphono-propionyl) piperazine-1-carboxylic, processes for their preparation, pharmaceutical compositions comprising said crystalline forms, pharmaceutical compositions prepared from such crystalline forms and their use as a medicament, especially as a p2y12 receptor antagonist.a invenção refere-se às formas cristalinas de cloridrato de éster butílico de ácido 4-((r)-2-{[6-((s)-3-metoxi-pirrolidin-1-il)-2-fenil-pirimidina-4 carbonil]-amino}-3-fosfono-propionil)-piperazina-1-carboxílico, processos para a preparação das mesmas, composições farmacêuticas compreendendo ditas formas cristalinas, composições farmacêuticas preparadas a partir de tais formas cristalinas e seu uso como um medicamento, especialmente como um antagonista do receptor p2y12.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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