CLEMENT, BERND,KOTTHAUS, JOSCHA,KOTTHAUS, JÜRKE,SCHADE, DENNIS
申请号：
EP11175252.3
公开号：
EP2550963A1
申请日:
2011.07.25
申请国别(地区):
EP
年份:
2013
代理人:
摘要：
Die vorliegende Erfindung betrifft Prodrug-Derivate des Pentamidins, ihre Verwendung zur Behandlung und/oder Prophylaxe von Krankheiten, insbesondere Tumorerkrankungen, sowie der Leishmaniose, Trypanosomiasis, der Pneumocystis carinii Pneumonie (PcP), sowie der Malaria.Pentamidine derivatives (I) are new. Pentamidine derivatives of formula (I) are new. n : 1-10. Independent claims are also included for: (1) salts, solvates and solvates of the salts of (I)； (2) a medicament comprising (I) and optionally at least one inert and non-toxic auxiliary； and (3) preparing (I). [Image] ACTIVITY : Cytostatic； Protozoacide； Antiinflammatory； Respiratory-Gen； Antimalarial. MECHANISM OF ACTION : None given.
