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AQUEOUS OPHTHALMIC SUSPENSION OF CRYSTALLINE REBAMIPIDE
专利权人:
发明人:
TAKAKUNI MATSUDA,SHOGO HIRAOKA,YUSO TOMOHIRA,SHINICHI ISHIKAWA
申请号:
MYPI 20055098
公开号:
MY152867A
申请日:
2005.10.28
申请国别(地区):
MY
年份:
2014
代理人:
摘要:
THE INVENTION PROVIDES AN OPHTHALMIC PRODUCT CONTAINING REBAMIPIDE, WHICH HAS A TRANSPARENCY ENOUGH TO BE AGREEABLE FEELING ON USING IT AND HAS NEUTRAL TO WEAKLY ACIDIC PH NOT TO INJURY OF THE KERATOCONJUNCTIVA OF A PATIENT SUFFERING FROM DRY EYE. AN AQUEOUS SUSPENSION OF CRYSTALLINE REBAMIPIDE WHICH HAS AN IMPROVED TRANSPARENCY IS PROVIDED BY ADDING AN AQUEOUS SOLUTION OF REBAMIPIDE DISSOLVED BY A BASE SUCH AS SODIUM HYDROXIDE OR AN AQUEOUS SOLUTION OF A SALT OF REBAMIPIDE TO AN AQUEOUS ACIDIC SOLUTION SUCH AS HYDROCHLORIC ACID CONTAINING AT LEAST ONE OF THE COMPOUNDS SELECTED FROM WATER-SOLUBLE POLYMERS AND SURFACTANTS, AND MIXING THEM. FIGURE 2
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