MCDERMOTT MICHAEL JAMES,JONAS MARCO,GAGE JENNIFER LYNN,BROT ELISABETH C A,LITTLE THOMAS L,CUTSHALL NEIL S,REINEKE KARL E,LUKE WAYNE DOUGLAS
申请号：
NZ63081014
公开号：
NZ630810A
申请日:
2014.09.10
申请国别(地区):
NZ
年份:
2016
代理人:
摘要：
Disclosed herein is a process for the preparation of compounds of Formula (II), which are useful in the inhibition of PDE10. In particular, the present invention is directed to an improved process for the preparation of 1-(5-(4-chloro-3,5-dimethoxyphenyl)furan-2-yl)-2-ethoxy-2-(4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl)ethanone, which is useful in the inhibition of PDE10.
