WILLMS, Lothar,SCHMITT, Monika H.,FRENZEL, Thomas,HAAF, Klaus Bernhard,HÄUSER-HAHN, Isolde,HEINEMANN, Ines,GATZWEILER, Elmar,ROSINGER, Christopher Hugh,DITTGEN, Jan,FEUCHT, Dieter,HILLS, Martin Jeffre
申请号:
ES12713928
公开号:
ES2612694T3
申请日:
2012.03.26
申请国别(地区):
ES
年份:
2017
代理人:
摘要:
3-Phenylisoxazolin-5-carboxamides and 3-phenylisoxazolin-5-thioamides of formula (I) or their salts ** Formula ** in which R1 and R2 independently mean each other hydrogen, fluorine, chlorine, bromine, iodine, cyano, or (C1-C4) alkyl or (C1-C4) alkoxy substituted respectively with m moieties of the group consisting of fluorine, chlorine, bromine, iodine and cyano, or R1 and R2 form together with the carbon atom to which they are attached a ring of three, four or five members saturated or partially or totally unsaturated, consisting of q carbon atoms and p oxygen atoms; R3 means fluorine, chlorine, cyano, (C1-C3) alkylcarbonyloxy or S (O) nR5, or (C1-C6) alkyl, cycloalkyl (C3-C6), alkenyl (C2-C6) or substituted (C2-C6) alkynyl respectively with m moieties of the group consisting of fluorine, chlorine, bromine, iodine, cyano, alkoxy (C1-C4) and hydroxy, or alkylcarbonyl (C1-C6), alkenylcarbonyl (C2-C6) or cycloalkylcarbonyl (C3-C6) substituted respectively with m residues of the group consisting of fluorine, chlorine, bromine, iodine, cyano and alkoxy (C1-C6); R4 means hydrogen, cyano, or (C1-C8) alkyl or cycloalkyl (C3-C8) substituted respectively with m moieties of the group consisting of fluorine, chlorine, bromine, iodine, cyano, hydroxy and (C1-C6) alkoxy; A means a bond or a divalent unit of the group consisting of ** Formula ** R10, R11, R12, R13, R14 and R15 each independently mean each other hydrogen, fluorine, chlorine, bromine, iodine, hydroxy, cyano, CO2R8, CONR6R8, R5, or (C1-C6) alkyl, cycloalkyl (C3-C5), alkenyl (C2-C6), alkynyl (C2-C6) substituted respectively with m moieties of the group consisting of fluorine, chlorine, bromine, iodine, hydroxy and cyano, or (C1-C6) alkoxy, cycloalkoxy (C3-C6), alkenyloxy (C2-C6) or alkynyloxy (C2-C6) substituted respectively with m moieties of the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2) alkoxy; And it means oxygen or sulfur; X means hydrogen, cyano, hydroxy, X1, or (C1-C12) alkyl,