PROCESS FOR SYNTHESIZING A CETP INHIBITOR

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专利权人:

Merck Sharp & Dohme Corp.

发明人:

COTE, Aaron S.,MILLER, Ross A.

申请号：

HK16101930.3

公开号：

HK1213815A

申请日:

2016.02.22

申请国别(地区):

HK

年份:

2016

代理人:

摘要：

An efficient process is disclosed for producing a compound that is an inhibitor of CETP. The last step of the process is the coupling of an oxazolidinone derivative with a biphenyl moiety to provide a compound of formula (I). In a specific embodiment of this synthesis, a crystalline product is produced which is characterized as a non-solvated crystalline polymorph.

来源网站：

中国工程科技知识中心

来源网址：

http://www.ckcest.cn/home/