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AZABICYCLIC CARBOXAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF
专利权人:
SANOFI-AVENTIS
发明人:
DUBOIS LAURENT,EVANNO, YANNICK,MACHNIK DAVID,MALANDA, ANDRÉ
申请号:
MYPI 2010003439
公开号:
MY150576A
申请日:
2009.01.20
申请国别(地区):
MY
年份:
2014
代理人:
摘要:
THE INVENTION RELATES TO THE COMPOUNDS OF GENERAL FORMULA (I) IN WHICH X₁, X₂, X₃ AND X₄ ARE, INDEPENDENTLY OF ONE ANOTHER, A NITROGEN ATOM OR A C-R₁ GROUP; Z₁, Z₂, Z₃ AND Z₄ ARE, INDEPENDENTLY OF ONE ANOTHER, A NITROGEN ATOM OR A C-R₂ GROUP; Ra AND Rb FORM, TOGETHER WITH THE CARBON ATOMS WHICH BEAR THEM, A FIVE-MEMBERED RING, THIS RING COMPRISING A NITROGEN ATOM AND CARBON ATOMS, THIS RING BEING PARTIALLY SATURATED OR UNSATURATED AND BEING OPTIONALLY SUBSTITUTED WITH ONE OR MORE SUBSTITUENTS R₃; W IS AN OXYGEN OR SULPHUR ATOM; n IS EQUAL TO 0, 1, 2 OR 3; Y IS AN OPTIONALLY SUBSTITUTED ARYL OR HETEROARYL; IN THE FORM OF A BASE OR OF AN ADDITION SALT WITH AN ACID, AND ALSO IN THE FORM OF A HYDRATE OR OF A SOLVATE. PROCESS FOR THE PREPARATION THEREOF AND THERAPEUTIC USE.
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