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SALTS OF AZA-BICYCLIC DI-ARYL ETHERS AND METHODS TO MAKE THEM OR THEIR PRECURSORS
专利权人:
NOVARTIS AG;노파르티스 아게
发明人:
MARTERER WOLFGANG,마터러, 볼프강,PRASHAD MAHAVIR,프라사드, 마하비르,VILLHAUER EDWIN BERNARD,빌하우어, 에드윈 버나드,WAYKOLE LILADHAR MURLIDHAR,웨이콜, 릴라드하르 멀리드하르,VIVELO JAMES ANTHONY,비벨로, 제임스 안토니,SUTTER BERTRAND,서터, 베르트랑,BIANC
申请号:
KR1020147003645
公开号:
KR1020140034309A
申请日:
2012.07.12
申请国别(地区):
KR
年份:
2014
代理人:
摘要:
The present invention relates to a process for the production of a compound of formula I ((R)-3-(6-(4-methylphenyl)-pyridin-3-yloxy)-1-aza-bicyclo[2.2.2]octane) or a salt thereof and to a process for the production of a compound of formula II (5-chloro-2-(4-methylphenyl)pyridine ) or a salt thereof, which is used as an intermediate in the preparation of the compound of formula I.본 발명은 (R)-3-(6-(4-메틸페닐)-피리딘-3-일옥시)-1-아자-비시클로[2.2.2]옥탄의 염, 상기 염 및 그의 전구체의 제조 방법, 그를 포함하는 제약 조성물, 및 의약으로서의 그의 용도에 관한 것이다.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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