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Substituted pyrimidin-4-one derivatives
专利权人:
サノフイ;田辺三菱製薬株式会社
发明人:
フアイヨル,オード,ロチード,アリステア,サデイ,ムラ,バツシユ,ジユリアン,イエシユ,フイリツプ,フアイヨル,オード,ロチード,アリステア,サデイ,ムラ,バツシユ,ジユリアン,イエシユ,フイリツプ
申请号:
JP2011515671
公开号:
JP5490790B2
申请日:
2009.06.25
申请国别(地区):
JP
年份:
2014
代理人:
摘要:
A pyrimidone derivative represented by formula (I) or a salt thereof, or a solvate thereof or a hydrate thereof: Y represents two hydrogen atoms, a sulphur atom, an oxygen atom, an hydroxy group and a hydrogen atom, an hydroxy group and a C 1-2 alkyl group, an hydroxy group and a C 1-2 perhalogenated alkyl group; a halogen atom and a hydrogen atom or a -(CH2)p-;Z represents a bond, an oxygen atom, NH, a nitrogen atom substituted by a hydrogen atom or a C 1-3 alkyl group, a sulphur atom, a methylene group optionally substituted ; R1 represents a 2, 3 or 4-pyridine ring or a 2, 4 or 5-pyrimidine ring, the ring being optionally substituted; R2 represents a hydrogen atom, a C 1-6 alkyl group or a halogen atom; R3 represents a hydrogen atom; a phenyl or a naphthyl group, these groups being optionally substituted a 4-15 membered heterocyclic group optionally substituted a -C(O)O (C 1-6 -alkyl) group optionally substituted ; a -C(O)-phenyl group, a -C(O)O-phenyl group, or a - C(O)O-CH 2 -phenyl group,the benzene rings of the above-mentioned groups being optionally substituted ; a -C(O)-4-15 membered heterocyclic group optionally substituted; R4 represents a hydrogen atom, a halogen atom, a hydroxyl group, a C 1-6 alkyl group optionally substituted; n represents 0 to 3; m represents 0 to 3 ; p represents 2 to 7; in the form of a free base or of an addition salt with an acid. Use in therapeutic
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