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AMINOINDAZOLE DERIVATIVES AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS INCLUDING THEM
专利权人:
AVENTIS PHARMA S.A.
发明人:
LESUISSE DOMINIQUE,DUTRUC-ROSSET GILLES,HALLEY FRANCK,BABIN DIDIER,ROONEY THOMAS
申请号:
MYPI 20033345
公开号:
MY146796A
申请日:
2003.09.04
申请国别(地区):
MY
年份:
2012
代理人:
摘要:
THE PRESENT INVENTION RELATES TO NOVEL DERIVATIVES OF GENERAL FORMULA (I) IN WHICH R3 IS A (1-6C) ALKYL, ARYL, ARYL(1-6C)ALKYL, HETEROARYL, HETEROARYL(1-6C)ALKYL, ARYL OR HETEROARYL FUSED TO A (1-10C)CYCLOALKYL, HETEROCYCLE, HETEROCYCLOALKYL, CYCLOALKYL, ADAMANTYL, POLYCYCLOALKYL, ALKENYL, ALKYNYL, CONR1R2, COOR1, SO2R1, C(=NH)R1 OR C(=NH)NR1 RADICAL; R5 AND R6 ARE, INDEPENDENTLY OF ONE ANOTHER, CHOSEN FROM THE FOLLOWING RADICALS: HALOGEN , CN, NO2, NH2, OH, COOH, C(O)OR8, —O—C(O)R8, NR8R9, NHC(O)R8, C(O)NR8R9, NHC(S)R8, C(S)NR8R9, SR8, S(O)R8, SO2 R8, NHSO2R8, SO2NR8R9, —O—SO2R8, —SO2—O—R8, TRIFLUOROMETHYL, TRIFLUOROMETHOXY, (1-6C)ALKYL, (1-6C)ALKOXY, ARYL , ARYL(1-6C) ALKYL, HETEROARYL, HETEROARYL(1-6C)ALKYL, HETEROCYCLE, CYCLOALKYL, ALKENYL, ALKYNYL, ADAMANTYL OR POLYCYCLOALKYL.
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中国工程科技知识中心
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