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专利权人:
ПРОКСИМАГЕН ЛИМИТЕД
发明人:
Дэвид,Эллисон,Элисон,Майкл,Эдвард,Айан,Марианне,Мартин,Эрик,Тобиас
申请号:
EA201490451
公开号:
EA201490451A1
申请日:
2011.09.14
申请国别(地区):
EA
年份:
2014
代理人:
摘要:
2- {4- [1- (4-Chlorophenyl) -1H-pyrrolo [2,3-c] pyridin-3-yl] piperidin-1-yl} ethan-1-amine; 3-aminopropyl 4- [1- (4-chlorophenyl) -1H-pyrrolo [2,3-c] pyridin-3-yl] piperidine-1-carboxylate; 1- {4- [1- (4-chlorophenyl) -1H-pyrrolo [2,3-c] pyridin-3-yl] piperidin-1-yl} -4- (dimethylamino) butan-1-one; 5-amino-1- {4- [1- (4-chlorophenyl) -1H-pyrrolo [2,3-c] pyridin-3-yl] piperidin-1-yl} pentan-1-one; N- (2-aminoethyl) -4- [1- (4-chlorophenyl) -1H-pyrrolo [2,3-c] pyridin-3-yl] piperidin-1-carboxamide; N- (3-aminopropyl) -4- [1- (4-chlorophenyl) -1H-pyrrolo [2,3-c] pyridin-3-yl] piperidin-1-carboxamide; 4- [1- (4-chlorophenyl) -1H-pyrrolo [2,3-c] pyridin-3-yl] -N- [3- (dimethylamino) propyl] piperidine-1-carboxamide; 1 - ({4- [1- (4-chlorophenyl) -1H-pyrrolo [2,3-c] pyridin-3-yl] piperidin-1-yl} carbonyl) piperazine; 4 - ({4- [1- (4-chlorophenyl) -1H-pyrrolo [2,3-c] pyridin-3-yl] piperidin-1-yl} carbonyl) morpholine; 1 - ({4- [1- (4-chlorophenyl) -1H-pyrrolo [2,3-c] pyridin-3-yl] piperidin-1-yl} carbonyl) -1,4-diazepan; ethyl 1- [1- (4-chlorophenyl) -1H-pyrazolo [3,4-c] pyridin-3-yl] piperidine-4-carboxylate; ethyl 1- [1- (4-methylphenyl) -1H-pyrazolo [3,4-c] pyridin-3-yl] piperidine-4-carboxylate; 1- [1- (4-chlorophenyl) -1H-pyrazolo [3,4-c] pyridin-3-yl] piperidin-4-carboxylic acid; N- (2-aminoethyl) -1- [1- (4-chlorophenyl) -1H-pyrazolo [3,4-c] pyridin-3-yl] piperidin-4-carboxamide; 4 - ({1- [1- (4-chlorophenyl) -1H-pyrazolo [3,4-c] pyridin-3-yl] piperidin-4-yl} carbonyl) morpholine; 1 - ({1- [1- (4-chlorophenyl) -1H-pyrazolo [3,4-c] pyridin-3-yl] piperidin-4-yl} carbonyl) piperazine; {4- [1- (4-methylphenyl) -1H-pyrazolo [3,4-c] pyridin-3-yl] morpholin-3-yl} methanol; {4- [1- (4-methylphenyl) -1H-pyrazolo [3,4-c] pyridin-3-yl] morpholin-2-yl} methanol; [(3R) -4- [1- (4-chlorophenyl) -1H-pyrazolo [3,4-c] pyridin-3-yl] morpholin-3-yl] methanol; methyl 4- [1- (4-chlorophenyl) -1H-pyrazolo [3,4-c] pyridin-3-yl] morpholine-3-carboxylate; N- (2-aminoethyl) -4- [1- (4-chlo
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