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quinoline and quinoxaline derivatives as protein tyrosine kinase inhibitors, their uses and manufacturing process, as well as pharmaceutical compositions and combinations comprising them
专利权人:
Novartis Ag
发明人:
Diana Graus Porta,Pascal Furet,Vito Guagnano
申请号:
BRPI0913031
公开号:
BRPI0913031A2
申请日:
2009.05.20
申请国别(地区):
BR
年份:
2019
代理人:
摘要:
Quinoline and quinoxaline derivatives as protein tyrosine kinase inhibitors The present invention relates to compounds of formula (I) wherein the substituents are as defined in the specification, in free form or in the form of a pharmaceutically acceptable salt, solvate, ester, n-oxide thereof; processes for their preparation; to pharmaceutical products containing such compounds, in particular for use in one or more protein tyrosine kinase mediated diseases.derivados de quinolina e quinoxalinas como inibidores de proteína tirosina quinase a presente invenção refere-se a compostos de fórmula (i) em que os substituintes são como definidos na especificação, na forma livre ou na forma de um sal farmaceuticamente aceitável, solvato, éster, n-óxido dos mesmos; processos para a preparação dos mesmos; a produtos farma-cêuticos contendo tais compostos, em particular para o uso em uma ou mais doenças mediadas por proteína tirosina quinase.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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