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PYRIDYLAMINOACETIC ACID COMPOUND AND POLYOXYETHYLENE CASTOR OIL-CONTAINING PHARMACEUTICAL COMPOSITION
专利权人:
САНТЭН ФАРМАСЬЮТИКАЛ КО., ЛТД.;SANTEN PHARMACEUTICAL CO., LTD.
发明人:
Yoko,Ёко
申请号:
EA201691139
公开号:
EA031723B1
申请日:
2015.01.08
申请国别(地区):
EA
年份:
2019
代理人:
摘要:
The purpose of the present invention is to provide a pharmaceutical composition that comprises (6{[4-(pyrazol-1-yl)benzyl](pyridine-3-ylsulfonyl)aminomethyl}pyridine-2-ylamino)isopropyl acetate or a salt thereof and polyoxyethylene castor oil, wherein the polyoxyethylene castor oil exhibits the number of polymerization of ethylene oxide in a range of 5 to 100, and wherein the content of the polyoxyethylene castor oil relative to (6{[4-(pyrazol-1-yl)benzyl](pyridine-3-ylsulfonyl)aminomethyl}pyridine-2-ylamino)isopropyl acetate or a salt thereof is in a range of 2/0.03 to 5,000 parts by mass relative to 1 part by mass of 6-{[4-(pyrazol-1-yl)benzyl](pyridin-3-ylsulfonyl)aminomethyl}pyridin-2-ylamino)isopropyl acetate or a salt thereof; and to provide a method for stabilizing (6-{[4-(pyrazol-1-yl)benzyl](pyridin-3-ylsulfonyl)aminomethyl}pyridin-2-ylamino)isopropyl acetate or a salt thereof by allowing a pharmaceutical composition comprising (6-{[4-(pyrazol-1-yl)benzyl](pyridin-3-ylsulfonyl)aminomethyl}pyridin-2-ylamino)isopropyl acetate or a salt thereof to comprise polyoxyethylene castor oil, wherein the polyoxyethylene castor oil exhibits the number of polymerization of ethylene oxide in a range of 5 to 100, and wherein the content of the polyoxyethylene castor oil relative to (6{[4-(pyrazol-1-yl)benzyl](pyridine-3-ylsulfonyl)aminomethyl}pyridine-2-ylamino)isopropyl acetate or a salt thereof is in a range of 2/0.03 to 5,000 parts by mass relative to 1 part by mass of 6-{[4-(pyrazol-1-yl)benzyl](pyridin-3-ylsulfonyl)aminomethyl}pyridin-2-ylamino)isopropyl acetate or a salt thereof.Цель настоящего изобретения заключается в обеспечении фармацевтической композиции, которая содержит (6-{[4-(пиразол-1-ил)бензил](пиридин-3-илсульфонил)аминометил}пиридин-2-иламино)изопропилацетат или его соль и полиоксиэтиленовое касторовое масло, где полиоксиэтиленовое касторовое масло имеет показатель полимеризации окиси этилена в диапазоне от 5 до 100 и где содержание полиоксиэтиленового к
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/
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