您的位置: 首页 > 农业专利 > 详情页

PYRROLIDIN-2-ONE DERIVATIVES AS ANDROGEN RECEPTOR MODULATOR
专利权人:
TAKEDA PHARMACEUTICAL COMPANY LIMITED
发明人:
HASUOKA, ATSUSHI
申请号:
MYPI 2010000564
公开号:
MY159910A
申请日:
2008.08.06
申请国别(地区):
MY
年份:
2017
代理人:
摘要:
A COMPOUND REPRESENTED BY THE FORMULA (I) WHERE IN R1 IS A HYDROGEN ATOM, A HALOGEN ATOM, A GROUP VIA A CARBON ATOM,A GROUP VIA A NITROGEN ATOM, A GROUP VIA AN OXYGEN ATOM OR A GROUP VIA A SULFUR ATOM;R2 IS A HYDROGEN ATOM, A HALOGEN ATOM, A GROUP VIA A CARBON ATOM, A GROUP VIA A NITROGEN ATOM, A GROUP VIA AN OXYGEN ATOM OR A GROUP VIA A SULFUR ATOM;R3 IS AN ELECTRON-WITHDRAWING GROUP; R4 IS A HYDROGEN ATOM, A HALOGEN ATOM, A GROUP VIA A CARBON ATOM, A GROUP VIA A NITROGEN ATOM, A GROUP VIA AN OXYGEN ATOM OR A GROUP VIA A SULFUR ATOM;R5 IS A HYDROGEN ATOM, A HALOGEN ATOM, A GROUP VIA A CARBON ATOM,A GROUP VIA A NITROGEN ATOM, A GROUP VIA AN OXYGEN ATOM OR A GROUP VIA A SULFUR ATOM;R6 IS A HYDROGEN ATOM, A HALOGEN ATOM, A GROUP VIA A CARBON ATOM,A GROUP VIA A NITROGEN ATOM, A GROUP VIA AN OXYGEN ATOM OR A GROUP VIA A SULFUR ATOM;R7 IS AN ALKYL GROUP OPTIONALLY HAVING SUBSTITUENT(S) OR AN ARALKYL GROUP OPTIONALLY HAVING SUBSTITUENT (S);R8 IS A HYDROGEN ATOM, AN ALKYL GROUP OPTIONALLY HAVING SUBSTITUENT (S), AN ALKENYL GROUP OPTIONALLY HAVING SUBSTITUENT(S) OR A CYCLOALKYL GROUP OPTIONALLY HAVING SUBSTITUENTS (S);R9 IS A GROUP VIA AN OXYGEN ATOM; AND RING A IS A 5- OR 6-MEMBERED RING OPTIONALLY FURTHER HAVING SUBSTITUENT(S) (IN THIS CASE, RING A MAY BE A 5- OR 6-MEMBERED RING FORMING A SPIRO BOND WITH C3-6 CYCLOALKANE), OR A SALT THEREOF HAS A SUPERIOR ANDROGEN RECEPTOR MODULATING ACTION.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充