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STABLE CRYSTAL FORM OF TIPIRACIL HYDROCHLORIDE AND CRYSTALLIZATION METHOD FOR THE SAME
专利权人:
TAIHO PHARMACEUTICAL CO.; LTD.
发明人:
KAZUNO, HIDEKI,MUTSUMI, TOMONOBU
申请号:
PH12015502809
公开号:
PH12015502809A1
申请日:
2015.12.17
申请国别(地区):
PH
年份:
2016
代理人:
摘要:
The present invention addresses the problem of producing a stabilized crystal of 5-chloro-6-[(2- iminopyrrolidin-1-yl)methyl]pyrimidine-2,4(1H,3H)-dione monohydrochloride. As a means for solving the problem, a crystal of 5-chloro-6-[(2-iminopyrrolidin-1-yl)methyl]pyrimidine-2,4(1H,3H)-dione monohydrochloride is provided. The crystal has characteristic peaks at diffraction angles (2? + 0.1o) of 11.6o, 17.2o, 17.8o, 23.3o, 27.1o and 29.3o in powder X-ray diffraction.
来源网站:
中国工程科技知识中心
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http://www.ckcest.cn/home/

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