The present invention relates to substituted benzo-pyrido-triazolo-diazepine compounds and methods of synthesizing these compounds. The present invention also relates to pharmaceutical compositions containing substituted benzo-pyrido-triazolo-diazepine compounds and methods of treating cell proliferative disorders, such as cancer, by administering these compounds or pharmaceutical compositions to subjects in need thereof.本發明係關於經取代的苯並-吡啶並-三唑並-二氮呯類化合物和合成這些化合物之方法。本發明亦關於含有經取代的苯並-吡啶並-三唑並-二氮呯類化合物的醫藥組成物和治療細胞增生性病症如癌症之方法,係藉由將這些化合物或醫藥組成物投予至需要其之個體。