Alan David Borthwick;Deirdre Mary Bernadette Hickey;Andrew McMurtrie Mason;John Liddle
发明人:
Alan David Borthwick,Deirdre Mary Bernadette Hickey,John Liddle,Andrew McMurtrie Mason
申请号：
US13035366
公开号：
US08202864B2
申请日:
2011.02.25
申请国别(地区):
US
年份:
2012
代理人:
摘要：
Compounds of formula (I)wherein R1 is 2-indanyl, R2 is 1-methylpropyl, R3 is a group selected from 2,6-dimethyl-3-pyridyl or 4,6-dimethyl-3-pyridyl, R4 represents methyl and R5 represents hydrogen or methyl or, R4 and R5 together with the nitrogen atom to which they are attached represent morpholino and pharmaceutically acceptable derivatives thereof are described, as are for their preparation, pharmaceutical compositions containing them and their use in medicine, particularly their use as oxytocin antagonists.
