MERCK PATENT GESELLSCHAFT MIT BESCHRÄNKTER HAFTUNG
发明人:
MARGARITA DRA. WUCHERER-PLIETKER,DANIELA DRA. WERKMANN,ANNE DRA. GIGOUT,DANIEL DR. KUHN,EDGAR SAWATZKY
申请号：
ARP130103053
公开号：
AR092266A1
申请日:
2013.08.28
申请国别(地区):
AR
年份:
2015
代理人:
摘要：
Claim 1: compounds of the formula (1), where W is n, or, ch u2082, ch u2082ch u2082, ch u2082choh (OR - or - ch u2082)； X, y, Q, u, T, independent of each other, c or n, provided that one or more of X, and q u and T, are carbon Atoms and M is linked to a carbon Atom； V is a link Simple cr u2074r u2075 or - or - or - M is cr u2074r u2075 - r u00b9 is heteroaryl,；Heterociclilo or mono - or bicyclic aryl containing 3 to 14 carbon Atoms and 1 or 4 heteroatoms selected independently of N, o and S, which is not replaced or is mono -, di - or trisustituido with r u2076； R u00b2 is H, a, CN, o oa or Hal； r u00b3 it is heterociclilo aryl or heteroaryl, Mono and bicyclic containing 3 to 14 carbon Atoms and 1 or 4 heteroatoms,Selected independently of N, o and S, which is not replaced or is mono -, di - or trisustituido with r u2077； r u2074, r u2075 are selected independently between themselves, the group consisting of H and r u2076； R u00b2, and r u2077 are selected independently of each other. Gr Upo is H, a, = o, Oh, OA, Hal (HAL) u2082 ch u2082hai, CH, C (HAL) u2083, no u2082 (ch u2082) u2099cn (ch u2082) u2099nr u2078r u2079 (ch u2082) u2099o ( u2096nr u2078r u2079, ch u2082)(ch u2082) u2099nr u2078 (ch u2082) u2096nr u2078r u2079 (ch u2082) u2099o (ch u2082) u2096or u00b9 u2078 (ch u2082) u2099nr u2078 (ch u2082) u2096or u2079 (ch u2082) u2099coor u00b9 u2070 (ch u2082) u2099chor u00b9 u2070, u2099chonr u2078r u2079 (ch u2082), C (o) C (o) nr u2078r u2079, nhanh u2082 (ch u2082) u2099nr u2078cor u00b9 u2070 ( u2099nr u2078conr u2078r u2079, ch u2082) (ch u2082) u2099nr u2078so u2082a (ch u2082 u2099so u2082nr u2078r u2079 (CH) u2082 u2099s () or () u1d58r u00b9 u2070, ch u2082 u2099oc () or () r u00b9 u2070, ch u2082 u2099c () or () r u00b9 u2070, ch u2082) u2099sr u2078, CH = n = N - ch u2082ch OA, OA, u2099nhoa (ch u2082), (ch u2082) u2099ch = N - r u2078 (ch u2082) u2099oc (OR) nr u2078r u2079 (ch u2082) u2099nr u2078coor u00b9 u2070 (ch u2
