GIJSEN, HENRICUS, JACOBUS, MARIA,OEHLRICH, DANIEL,BISCHOFF, FRANÇOIS PAUL,ZHUANG, WEI,VAN BRANDT, SVEN FRANCISCUS ANNA,SURKYN, MICHEL,ZAJA, MIRKO,BERTHELOT, DIDIER, JEAN-CLAUDE,DE CLEYN, MICHEL ANNA J
申请号：
MYPI 2011003788
公开号：
MY151983A
申请日:
2010.02.15
申请国别(地区):
MY
年份:
2014
代理人:
摘要：
THE PRESENT INVENTION IS CONCERNED WITH NOVEL SUBSTITUTED BENZOXAZOLE, BENZIMIDAZOLE, OXAZOLOPYRIDINE AND IMIDAZOPYRIDINE DERIVATIVES OF FORMULA (I) WHEREIN R1, R2, R3, R4, X, A1, A2, A3, A4, Y1, Y2, Y3 AND Z HAVE THE MEANING DEFINED IN THE CLAIMS. THE COMPOUNDS ACCORDING TO THE PRESENT INVENTION ARE USEFUL AS GAMMA SECRETASE MODULATORS. THE INVENTION FURTHER RELATES TO PROCESSES FOR PREPARING SUCH NOVEL COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAID COMPOUNDS AS AN ACTIVE INGREDIENT AS WELL AS THE USE OF SAID COMPOUNDS AS A MEDICAMENT. (NO SUITABLE FIGURE)
