CHRISTIAN LOTHSCHUETZ,HELMARS SMITS,MIROSLAV TERINEK,TOMAS SMEJKAL
申请号:
BR112016025076
公开号:
BR112016025076A2
申请日:
2015.04.30
申请国别(地区):
BR
年份:
2018
代理人:
摘要:
The present invention relates to processes for the preparation of substituted cycloserine compounds of formula (I) wherein R1 is C1-C8alkyl, C1-C8haloalkyl, C3-C6cycloalkyl, aryl or aryl substituted by one to five R11, or aryl-C1-C4alkylene or aryl-C1-C4alkylene substituted by one to five R11; and each R11 is independently C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy, cyano or halogen; The invention also relates to intermediates produced by the processes. Compounds of formula (I) are useful intermediates for the production of compounds in the agricultural and pharmaceutical fields.