ITOH, TETSUJI,JEON, INGYU,MANGION, IAN,QIAN, GANG,SHERRY, BENJAMIN, D.,GAUTHIER, DONALD, R.,CAO, YANG
申请号:
EP13860921
公开号:
EP2928472A4
申请日:
2013.12.04
申请国别(地区):
EP
年份:
2016
代理人:
摘要:
The present invention is directed to a novel process for synthesizing 3-(substituted phenoxy)-1-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl])-pyridin-2(1H)-one derivatives. The compounds synthesized by the processes of the invention are HIV reverse transcriptase inhibitors useful for inhibiting reverse transcriptase, HIV replication and the treatment of human immunodeficiency virus infection in humans.