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OIL-BASED PREPARATION CONTAINING ANTIPROTOZOAL TRIAZINES AND ANTHELMINTIC CYCLODEPSIPEPTIDES
专利权人:
发明人:
申请号:
HK17100321.1
公开号:
HK1226657A
申请日:
2017.01.11
申请国别(地区):
HK
年份:
2017
代理人:
摘要:
This refers to a preparation comprising a triazine based Oil that is active against parasitic protozoa and a cyclodepsipeptide Vermifuge, Preparation is particularly suitable for oral Application of the combination of active substances in animals.Claim 1: preparations comprising a triazine is active against parasitic Protozoa, and have a particle size D (90) < = 15 mm and a cyclodepsipeptide Vermifuge in an oil base.Claim 2: preparation according to claim 1, in which the triazine is a compound of the formula (1) or (2) in which R1 R3 represents - SO2 - or - S - R3, R2 is alkyl, alkoxy, halogen or so2n (CH3) 2 and represents haloalquilo R3, R4 and R5 independently one another represent IC and R6 represents Hydrogen or Fluorine or chlorine, and their physiologically acceptable Salts.Claim 3: preparation according to one of the preceding Claims, in which the diclazuril, toltrazuril ponazuril triazine is, or. Claim 2: preparation according to claim 4, in which the cyclic depsipeptide PF is 1022. Preparation according to claim 7: one of the preceding Claims, comprising in particular a Thickener, a glycerol Ester.Claim 1: Use of Preparations according to one of the preceding claims for the preparation of pharmaceutical products for controlling parasitic protozoa and endoparasites in humans or animals.La presente se refiere a una preparacion basada en aceite que comprende una triazina que es activa contra protozoos parásitos y un ciclodepsipéptido vermífugo, preparacion que es particularmente adecuada para la aplicacion oral de la combinacion de sustancias activas en animales. Reivindicacion 1: Preparaciones que comprenden una triazina que es activa contra protozoos parásitos y tiene un tamano de partícula d(90) <= 15 mm y un ciclodepsipéptido vermífugo en una base de aceite. Reivindicacion 2: Preparacion segun la reivindicacion 1, en la que la triazina es un compuesto de las formulas (1) o (2) en las que R1 representa R3-SO2- o R3-S-, R2 representa alquilo, alcoxi, haloge
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