트리아진 유도체의 신규한 의학적 용도
- 专利权人:
- 发明人:
- 리치, 마이클,하르비지, 로렌스,리달, 디에테르,바라클로지, 파울
- 申请号:
- KR1020097002878
- 公开号:
- KR1014820490000B1
- 申请日:
- 2007.07.13
- 申请国别(地区):
- KR
- 年份:
- 2015
- 代理人:
- 摘要:
- Compounds of formula (I) especially where R1 is an optionally substituted alkyl, aralkyl or heterocyclyl-alkyl group, are shown to have activity as sodium channel blockers or as antifolates. Some novel compounds where R1 is an aralkyl or heterocyclyl-alkyl are disclosed.화학식 I특히, R1이 선택적으로 치환된 알킬, 아르알킬 또는 헤테로사이클릴-알킬 기인 화학식 (I) 화합물은 나트륨 채널(sodium channel) 차단제(blocker)로서 또는 항엽산제(antifolate)로서 활성을 갖는 것으로 밝혀졌다. R1이 아르알킬 또는 헤테로사이클릴-알킬인 일부 신규한 화합물이 개시된다.
- 来源网站:
- 中国工程科技知识中心
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