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HETEROCYCLIC COMPOUND AND PHARMACEUTICAL COMPOSITION THEREOF
专利权人:
OTSUKA PHARMACEUTICAL CO.; LTD.
发明人:
SUMIDA, TAKUMI,TABUSA, FUJIO,SEKIGUCHI, KAZUO,KODAMA, TAKESHI,YASUMURA, KOICHI,KOJIMA, YUTAKA,MOTOYAMA, MASAAKI,MIYAJIMA, KEISUKE,YOSHIDA, KENJI,KAN, KEIZO,SAKAMOTO, MAKOTO,TAKASU, HIDEKI,NAKAGAWA, TA
申请号:
NZ58457308
公开号:
NZ584573A
申请日:
2008.10.29
申请国别(地区):
NZ
年份:
2012
代理人:
摘要:
Disclosed are heterocyclic compounds, or salts thereof, represented by general formula (I). Examples of the heterocyclic compound include: N-Dimethyl-M-[6-(2-{ 4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl} -1H-indol-6-yloxy)pyridin-3-yl]benzenesulfonamide, 3,4-Dichloro-N-(2-{ 2-[4-(4-isopropoxybenzyl)piperazine-1-carbonyl]-1-methyl-1H-indol-6-yloxy} pyrimidin-5-yl)-N-methylbenzenesulfonamide, and N-[6-(2-(4-[(4-Methoxybenzyl)methylamino]piperidine-1-carbonyll-1-methyl-1H-indol-5-yloxy)pyridin-3-yl]-4-trifluoromethylbenzamide. The compounds are used to treat fibrosis and tumours.
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