OPIOID RECEPTOR MODULATORS AND USE THEREOF

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专利权人:

National Health Research Institutes;Regents of the University of Minnesota

发明人:

Shau-Hua Ueng,Shiu-Hwa Yeh,Horace Loh,Yu-Sheng Chao

申请号：

US15207951

公开号：

US20170056377A1

申请日:

2016.07.12

申请国别(地区):

US

年份:

2017

代理人:

摘要：

Disclosed is an in vitro screening method for identifying an antagonist-to-agonist allosteric modifier of a mu-opioid receptor and an in vivo method for confirming that a test compound is such a modifier of a mu-opioid receptor. Also disclosed is a method for treating an opioid receptor-associated condition using a compound of Formula (I) and a pharmaceutical composition containing the same.

来源网站：

中国工程科技知识中心

来源网址：

http://www.ckcest.cn/home/