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sphingosine kinase inhibitors
专利权人:
MERCK PATENT GMBH
发明人:
DIRK WIENKE,FRANK STIEBER
申请号:
BR112012014164
公开号:
BR112012014164A2
申请日:
2010.11.22
申请国别(地区):
BR
年份:
2016
代理人:
摘要:
sphingosine kinase inhibitors the present invention relates to compounds of formulaq (i) wherein r1, r2, r3, r4, r5, r6, r7, r8, r9, r10, r11, r12, r13, r14, r15, r16 , r17, m1, m2, m3, m4, y1, y2, v, w, n, and m have the meanings indicated in claim 1, and physiologically acceptable salts, derivatives, prodrugs, solvates, tautomers and stereoisomers thereof, including those their mixtures in all reasons for use in the treatment of diseases that are influenced by inhibition of sph kinase 1.inibidores da esfingosina quinase a presente invenção refere-se a compostos da fórmulaq (i) em que r1, r2, r3, r4, r5, r6, r7, r8, r9, r10, r11,r12, r13, r14, r15, r16, r17, m1, m2, m3, m4, y1, y2, v, w, n, m e o possuem os significados indicados na reivindicação 1, e sais fisiologicamente aceitáveis, derivados, pró-fármacos, solvatos, tautômeros e estereoisômeros desses, incluindo as suas misturas em todas as razões, para o uso no tratamento de doenças que são influenciadas pela inibição de sph quinase 1.
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