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Tetrahydropyridine Compounds
专利权人:
EISAI RandD MANAGEMENT CO.; LTD.
发明人:
BOIVIN, Roch,CARLSON, Eric,ENDO, Atsushi,HANSEN, Hans,ISHIZAKA, Sally,MACKEY, Matthew,NARAYAN, Sridhar,SATOH, Takashi,SCHILLER, Shawn,HAWKINS, Lynn D.
申请号:
PE2019000725
公开号:
PE20190973A1
申请日:
2013.05.31
申请国别(地区):
PE
年份:
2019
代理人:
摘要:
It is a method of treating lupus erythematosus, including effective drug management of a compound (4,5,6,7-tetrahydropyridine (1,5-A) in formula (I), in which R1 is an alternative pyridine and an alternative pyridine. IODA, 1,4-dimethylthiazole pyridine, etc; R7 ES-CF3 O-CHF2; R8 is 1,2-dimethoxybenzene or 1,3-dimethyl-1H-pyrazole; R9 is BR, CL, F, I or H. These compounds are cubic or alien to the receivers of TOLL (TLR) 7 and 8.SE REFIERE A UN METODO PARA EL TRATAMIENTO DE LUPUS ERITEMATOSO SISTEMICO QUE COMPRENDE ADMINISTRAR UNA CANTIDAD FARMACEUTICAMENTE EFICAZ DE UN COMPUESTO 4,5,6,7-TETRAHIDROPIRAZOLO[1,5-A]PIRIMIDINA DE FORMULA (I) DONDE R1 ES PIPERIDINILO OPCIONALMENTE SUSTITUIDO, PIRROLIDINILO OPCIONALMENTE SUSTITUIDO, 1,4-DIMETILTIAZOLILO, ENTRE OTROS; R7 ES -CF3 O -CHF2; R8 ES 1,2-DIMETOXIBENCENO O 1,3-DIMETIL-1H-PIRAZOL; R9 ES Br, Cl, F, I O H. DICHOS COMPUESTOS ACTUAN COMO ANTAGONISTAS O INIHIBIDORES DE LOS RECEPTORES SIMILARES A TOLL (TLR) 7 Y 8
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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