您的位置: 首页 > 农业专利 > 详情页

solid forms of a selective cdk4 / 6 inhibitor
专利权人:
PFIZER INC.
发明人:
BRIAN PATRICK CHEKAL,NATHAN D. IDE
申请号:
BR112015019508
公开号:
BR112015019508A8
申请日:
2014.02.08
申请国别(地区):
BR
年份:
2019
代理人:
摘要:
Summary "solid forms of a selective cdk4 / 6 inhibitor" This invention relates to the crystalline free base of acetyl-8-cyclopentyl-5-methyl-2- (5-piperazin-1-yl-pyridin-2-ylamino) - 8h-pyrido [2,3-d] pyrimidin-7-one which exhibits improved properties, to pharmaceutical compositions and dosage forms comprising the free base and methods for making and using such compounds, compositions and dosage forms in the treatment of diseases. proliferative cells, such as cancer.resumo “formas sólidas de um inibidor de cdk4/6 seletivo” esta invenção se refere à base livre cristalina de acetil-8-ciclopentil-5-metil-2-(5-piperazin-1-il-piridin-2-ilamino)-8h-pirido[2,3-d]pirimidin-7-ona que apresenta propriedades aperfeiçoadas, às composições farmacêuticas e formas de dosagem compreendendo a base livre e aos métodos para fabricar e usar tais compostos, composições e formas de dosagem no tratamento de doenças celulares proliferativas, tais como câncer.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充