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7-cyclopentadiene-2 - (5-piperazin-1-il-piridin-2-il-amino) - 7h-pirrolo - [2, 3-d] - pirimidin-6-carboxyl and process for elaboration
专利权人:
NOVARTIS AG;ASTEX THERAPEUTICS LIMITED
发明人:
KAPA PRASAD, KOTESWARA,GONG, BAOQING,CALIENNI, JOHN VINCENT,CHEN, GUANG-PEI,SAXENA, VISHAL
申请号:
ECSP13012619
公开号:
ECSP13012619A
申请日:
2013.05.10
申请国别(地区):
EC
年份:
2013
代理人:
摘要:
This Invention refers to: (1) a process for preparing Dimethyl acid amide ciclopentil - 7 - 2 - (5 - (piperazin-1-yl pyridin-2-yl - amino) - 7h pyrrolo [2,3-d] - pyrimidine - 6 - carboxylic acid and salts thereof; 2) New salts of Dimethyl acid amide ciclopentil - 7 - 2 - 5 - (piperazin-1-yl - pyridin-2-yl - Amin (o) - 7h pyrrolo [2,3 - d] pyrimidine carboxylic - 6 - (3); Pharmaceutical compositions comprising the same; and (4) Methods for treatment using the same.Esta invención se refiere a: (1) un proceso para elaborar dimetil-amida del ácido 7-ciclopentil-2-(5-piperazin-1-il-piridin-2-il-amino)-7H-pirrolo-[2,3-d]-pirimidin-6-carboxílico y sales de la misma; (2) sales nuevas de dimetil-amida del ácido 7-ciclopentil-2-(5-piperazin-1-il-piridin-2-il-amino)-7H-pirrolo-[2,3-d]-pirimidin-6-carboxílico; (3) composiciones farmacéuticas que comprenden la misma; y (4) métodos para el tratamiento utilizando la misma.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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