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Quinazolinicos derivatives useful for treating central nervous system Disorders and Pharmaceutical compositions containing them
专利权人:
OTSUKA PHARMACEUTICAL CO.; LTD.
发明人:
MASAKI SUZUKI,MUNEAKI KURIMURA,KRISHNA R. VALLURU,AKIRA TAKAHASHI,TAKESHI KURODA,HARUKA TAKAHASHI,TAE FUKUSHIMA,SHIN MIYAMURA,INDRANATH GHOSH,ABHISHEK DOGRA,GERALDINE HARRIMAN,AMY ELDER,SATOSHI SHIMIZ
申请号:
ARP120102337
公开号:
AR086798A1
申请日:
2012.06.28
申请国别(地区):
AR
年份:
2014
代理人:
摘要:
1. Requirement 1: a compound (1) with formula characteristics,Or salt, where m is 0 or 1, l is a direct link or n8310;R¹ is hydrogen, C₁₋₈ alkyl,Halogenated tar c83218c8331-8328;a. Alcox c832188331s 8328; rent c832188331s 8328;Calcium hydroxide c83216c83318328;C₁₋₈ aminoalkyl,oxazolilo tiazolilo isoxazolilo piridilo pirrolopiridilo oxadiazolilo-alquilo CPiridilo asphalt c8321c83318328;Oxazolilo asphalt c8321c 83318328;3. Phenyl-c83218c83318328;-C (O) Rpirrolidinilo azetidinilo indolinilo piperidinilo morfolinilo piperazinilo fenilo cicloalquilo CC₃₋₈ cycloalkyl C₁₋₈alkyl,1. Benzoxazolilo, each substance can be replaced by 1-2r8311;R² is C₁₋₈ alkoxy,1 Isoquinol, benzofuran, dihydrobenzofuran, benzodiazepine, dihydrobenzoxazinilo, dihydrobenzodiazepine, tetrahydrobenzoxazepinilo, isoindian forest, Indian forest, Tianjin or dihydrobenzodiazepine were selectively replaced by 1-3r8313;R³ is pyridyl, pyrimidinyl, pyrazinyl or pyridazinyl, each of which is optionally substituted with C₁₋₈ alkyl,C₁₋₈ alkoxy,halo, haloalkyl C₁₋₈,C₁₋₈ haloalkoxy,cyano or -ORᵈ;R⁴ is hydrogen, C₁₋₈ alkyl,C₁₋₈ alkoxy,halo, C₁₋₈ haloalkyl or C₁₋₈ haloalkoxy,Each alternative number is r83044;R⁶ is hydrogen or C₁₋₈ alkyl;R⁷ is C₁₋₈ alkyl,C₂₋₈ alkenyl,1. C 83228331 asphalt;Arilo, heateral, ccilo, heatcycle, arilalquilo, heateral lalquilo, ccilalquilo, heatcycleo, halo, haloteoqui, hailoalcoxi, amino quilo, rented tar, diallaminoquile, hydroxil quilo, alcoquilo, alcoxie, oxo, tioxo CN, - no832222;-C (O) OR-C (y) 7495; (r74955,-No. 7580; (C (y) r758080;No. 7495; r74955,-OC (O) NR R-No. 7580; - No. C (o) 758080;-So8322; - No. 749595; - r74955;-No. 7580; - No. so8322; - No. 758080;-No. 7580; (C (y) No. 7495; r74955;-Or74966,-74966,-C (Y) R o S (O) qR1. Each alternative is replaced by R2;R⁹ is C₁₋₈ alkyl,C₁₋₈ alkoxy,1. Phenyl, PYRAZOLIN, dihydrobenzoxazolilo, oxazolilo, tetrazolilo, pyridazole Lilo, tiazolyl lo, cyclopentaaurol c83231;oxetanilo pirrolidinilo morfolinilo halo haloalquilo CC₁₋₈ haloalkoxy,
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/
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