Zhe Nie,Jeffrey Alan Stafford,James Marvin Veal,Michael Brennen Wallace
申请号:
US14098415
公开号:
US08987461B2
申请日:
2013.12.05
申请国别(地区):
US
年份:
2015
代理人:
摘要:
Provided herein are substituted pyrazolylpyridine, pyrazolylpyridazine, and pyrazolylpyrimidine derivative compounds and pharmaceutical compositions comprising said compounds. The subject compounds and compositions are useful for inhibition histone demethylase. Furthermore, the subject compounds and compositions are useful for the treatment of cancer, such as prostate cancer, breast cancer, bladder cancer, lung cancer and/or melanoma and the like.