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SNAR PROCESS FOR PREPARING BENZIMIDAZOLE COMPOUNDS
专利权人:
发明人:
DEMATTEI JOHN,BARNETT BRADLEY R.,LEONARD JOHN,SHAKYA SAGAR,NICHOLS PAUL J.,HACHE BRUNO P.,EVANS MATTHEW CHARLES,FORD JAMES GAIR
申请号:
IN9781/DELNP/2007
公开号:
IN270067B
申请日:
2007.12.17
申请国别(地区):
IN
年份:
2015
代理人:
摘要:
Provided are methods for the synthesis of heterocyclic compounds such as benzimidazole carboxylic acid core structures having Formula Ia-2 and their synthetic intermediates: wherein X1, X2, X5, R1, R2 and R4 are as defined herein. Compounds of Formula Ia-2 and their synthetic intermediates can be used to prepare heterocyclic derivatives such as benzimidazole derivatives.
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