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Crystalline form of 2-tiyazoril-4-quinine-o derivative, a powerful hexachlorobenzene inhibitor
专利权人:
BOEHRINGER INGELHEIM INTERNATIONAL GMBH
发明人:
BERKENBUSCH, THILO,BUSSACA, CARL ALAN,JAEGER, BURKHARD,VARSOLONA, RICHARD J.
申请号:
PE2012002419
公开号:
PE20130307A1
申请日:
2009.09.14
申请国别(地区):
PE
年份:
2013
代理人:
摘要:
It refers to a crystal sodium salt. Its derivative is 2-tiazolil-4-quinolini-oxi (1), which contains an X-ray powder derivative. Its peak value is 5.4, 6.5, 8.7, 10.1, 11.9, 13.0, 18.2, 20.2 and 24.7 ° 2teta. It is measured by cuka radiation. He also mentioned a pharmaceutical composer These compounds are enzyme inhibitors of hepatitis C virus and effective tools for the treatment of hepatitis C virus infection.SE REFIERE A UNA SAL DE SODIO CRISTALINA DE UN DERIVADO DE 2-TIAZOLIL-4-QUINOLINIL-OXI DE FORMULA (1) QUE TIENE UN PATRON DE DIFRACCION DE RAYOS X EN POLVO QUE COMPRENDE PICOS A 5,4; 6,5; 8,7; 10,1; 11,9; 13,0; 18,2; 20,2 Y 24,7 GRADOS 2THETA CUANDO SE MIDE USANDO RADIACION CuKa. TAMBIEN SE REFIERE A UNA COMPOSICION FARMACEUTICA. DICHOS COMPUESTOS SON INHIBIDORES DE LA SERINA PROTEASA NS3 DEL VIRUS DE LA HEPATITIS C SIENDO UTILES EN EL TRATAMIENTO DE INFECCIONES CAUSADAS POR EL VIRUS DE LA HEPATITIS C
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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