JIANG ROBERT H.,ZABLOCKI JEFF,CHIN GREGORY,AKTOUDIANAKIS EVANGELOS,CORKEY BRITTON KENNETH,DU JINFA,ELBEL KRISTYNA,KOBAYASHI TETSUYA,MARTINEZ RUBEN,METOBO SAMUEL E.,MISH MICHAEL,SHEVICK SOPHIE,SPERANDI
申请号:
NZ71158614
公开号:
NZ711586A
申请日:
2014.03.27
申请国别(地区):
NZ
年份:
2016
代理人:
摘要:
This application relates to chemical compounds which may act as inhibitors of, or which may otherwise modulate the activity of, a bromodomain-containing protein, including bromodomain-containing protein 4 (BRD4), and to compositions and formulations containing such compounds, and methods of using and making such compounds. Compounds include compounds of Formula (I) wherein R1a, R1b, R2a, R2b, R3, and X are described herein.